BASAVARAJAIAH S M | Medicinal Chemistry | Best Researcher Award

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Dr. BASAVARAJAIAH S M | Medicinal Chemistry | Best Researcher Award

Assistant Pfessorro, Vijaya College, Bangalore

Dr. Basavaraijaiah S. M. is an accomplished chemist with 15 years of teaching and industrial research experience. He has published extensively in national and international journals, authored books, book chapters, and holds patents. Currently, he serves as Coordinator of the P.G. Department of Chemistry at Vijaya College, Bangalore. He has held positions as an Assistant Professor and Principal Scientist in leading institutions and industries. His research focuses on the synthesis and biological activities of heterocyclic compounds. Recognized globally, he is among Stanford University’s Top 2% Scientists (2024). He is an editorial board member for several reputed journals, including Discover Applied Sciences and Journal of Chemistry. Dr. Basavaraijaiah has guided numerous postgraduate students and successfully led funded research projects. He actively organizes national and international chemistry conferences and serves as a BOS and BOE member for various universities, contributing significantly to chemical sciences and education.

Scholar

profile

🎓 Education 

Dr. Basavaraijaiah S. M. holds a Ph.D. in Chemistry (2009) from Gulbarga University, specializing in the synthesis and biological activities of heterocyclic compounds. He completed his M.Sc. in Chemistry (2004) from the same institution and earned his B.Sc. (2002) from Kottureshwara College, Karnataka. His academic journey laid the foundation for his expertise in organic synthesis and medicinal chemistry. Throughout his education, he developed a strong research aptitude, which later led to significant contributions in chemistry through publications, patents, and research projects. His doctoral research focused on nitrogen, oxygen, and sulfur-containing heterocycles, advancing knowledge in pharmaceutical chemistry. Postdoctoral studies at IIT Kanpur further refined his expertise. His academic credentials and continuous learning have positioned him as an authority in chemical sciences, mentoring students and advancing research in organic chemistry.

💼 Experience 

Dr. Basavaraijaiah S. M. has held key academic and industrial positions, currently serving as Coordinator of the P.G. Department of Chemistry at Vijaya College, Bangalore (since 2017). Previously, he was an Assistant Professor at the same institution (2014-2017). His industry experience includes roles as Principal Scientist at Skanda Life Sciences (2013-2014), Senior Scientist (2011-2013), and Group Leader (2010-2011) at LGC Promochem India Pvt. Ltd. He was a Postdoctoral Fellow at IIT Kanpur (2009-2010), enhancing his research in organic chemistry. Earlier, he worked as a Guest Lecturer at Gulbarga University (2007-2008) and as a Trainee Chemist at VB Medicare Pvt. Ltd. (2004-2005). His diverse career integrates academic excellence with industrial applications, contributing to education, research, and scientific advancements.

🏆 Awards & Honors

Dr. Basavaraijaiah S. M. has received global recognition, including being listed among Stanford University’s Top 2% Scientists (2024). His research has earned an H-index of 20 with over 1,400 citations. He has secured multiple grants, including VGST-SPICE funding (2015-16) and a UGC Minor Research Project (₹5 lakh, 2016-2018). He has guided 25 postgraduate students in research and successfully organized several national and international chemistry webinars and workshops. His editorial roles include serving on the boards of Discover Applied Sciences (Springer), Journal of Chemistry (Wiley), and Arkivoc Journal (Arkat USA). Additionally, he is an editorial advisor for Cambridge Scholars Publishing, UK. His contributions to chemical sciences, education, and research have made a significant impact, establishing him as a leader in his field.

🔬 Research Focus

Dr. Basavaraijaiah S. M.’s research focuses on the synthesis and biological activities of heterocyclic compounds, particularly nitrogen, oxygen, and sulfur-based derivatives. His work explores medicinal chemistry applications, aiming to develop novel therapeutic agents. He is actively involved in organic synthesis, green chemistry, and catalytic processes. His contributions extend to drug discovery, material sciences, and sustainable chemistry. He has authored numerous high-impact publications, patents, and book chapters, advancing knowledge in pharmaceutical and industrial chemistry. His research collaborations include academia and industry, fostering innovation in chemical sciences. His expertise in heterocyclic synthesis has led to significant developments in bioactive compounds with potential pharmaceutical applications. He continues to mentor postgraduate students and engage in cutting-edge research, pushing the boundaries of chemistry.

Conclusion

Dr. Basavaraiaiah S. M. is a highly qualified and accomplished researcher with strong credentials in academia, research, and editorial roles. His global recognition, project funding, and research impact make him a strong contender for the Best Researcher Award. Strengthening industry collaborations, international partnerships, and high-impact publications could further solidify his candidacy.

publication

Title: Therapeutic potential of pyrrole and pyrrolidine analogs: an update
Author(s): N Jeelan Basha, S M Basavarajaiah, K Shyamsunder
Year: 2022
Citation: 126

Title: A comprehensive insight on the biological potential of embelin and its derivatives
Author(s): N J Basha, S M Basavarajaiah, S Baskaran
Year: 2022
Citation: 38

Title: Exploration of Indolo [3, 2c] isoquinoline derived triazoles as potential antimicrobial and DNA cleavage agents: synthesis, DFT calculations, and molecular modeling
Author(s): S M Basavarajaiah, J Badiger, N G Yernale, N Gupta
Year: 2023
Citation: 21

Title: Synthesis, spectral analysis, DFT calculations, biological potential and molecular docking studies of indole appended pyrazolo-triazine
Author(s): S M Basavarajaiah, G Y Nagesh, M Javeed, R Bhat
Year: 2023
Citation: 31

Title: Anticancer potential of bioactive molecule luteolin and its analogs: An update
Author(s): N J Basha, S M Basavarajaiah
Year: 2023
Citation: 18

Title: Investigating the molecular interactions of 11-substituted-1-(4-chlorophenyl)-8H-indolo [3, 2-c][1, 2, 4] triazolo [3, 4-a] isoquinolines for Antimicrobial Potential
Author(s): M Ahmed, R Nalini, S M Basavarajaiah
Year: 2024
Citation: 6

Title: Naphtho [2, 1-b] furan derived triazole-pyrimidines as highly potential InhA and Cytochrome c peroxidase inhibitors: synthesis, DFT calculations, drug-likeness profile
Author(s): K S Kiran, M Selvaraj, S M Basavarajaiah
Year: 2023
Citation: 21

 

Nozuko Blasich | HIV and Mycology | Best Researcher Award

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Ms. Nozuko Blasich | HIV and Mycology | Best Researcher Award

Quality Control Technologist, National Health Laboratory Service South Africa

Nozuko Blasich is a Clinical Pathology Medical Technologist specializing in laboratory diagnostics, quality control, and biomedical research. She holds a Master of Science in Biomedical Technology and is currently pursuing a PhD in Biomedical Science, focusing on fungal pathogens and their public health impact. Her research on cryptococcal meningitis has influenced World Health Organization (WHO) policies. She has published in high-impact journals, presented at international conferences, and serves as a peer reviewer. Passionate about improving diagnostic accuracy, she explores point-of-care tests for infectious diseases.

Profile

Orcid

Education 🎓

Nozuko Blasich earned her Master of Science in Biomedical Technology, with research focusing on cryptococcal meningitis, significantly contributing to global health policies. She is currently a PhD candidate in Biomedical Science, investigating fungal pathogens and their environmental prevalence. Her academic journey emphasizes microbiology, clinical diagnostics, and public health.

Experience 🧑‍🏫

She serves as a Quality Control Technologist at the National Health Laboratory Service, ensuring diagnostic accuracy and laboratory efficiency. With expertise in mycology, she has worked extensively on cryptococcal antigen screening and HIV diagnostics.

 Awards & Honors 🏆

She has received recognition for her contributions to medical mycology, including best researcher awards and grants for her impactful studies on fungal pathogens and diagnostic advancements.

Research Interests 🔬

Her research explores fungal infections, laboratory diagnostics, and point-of-care testing to enhance public health interventions. She investigates diagnostic methodologies, antimicrobial resistance, and epidemiology to improve early detection and treatment outcomes.

Publications 📚

  1. Evaluating the Accuracy of Multiple Rapid Diagnostic Tests for HIV Detection in Serum Samples Analysed During Point-of-Care Proficiency Testing Assessments (2025) – Nozuko P. Blasich, Jerom Okot, Artur Ramos, Mduduzi B. Buthelezi, Dumisani F. Shabangu, Mahlatse M. Maleka, Sarvashni Moodliar, Nqobile Ngoma, Tendesayi Kufa

 

  1. Retrospective Assessment of a National Reflex Cryptococcal Antigen Screening Program in South Africa Through Interlaboratory Comparison of Lateral Flow Assay Results (2022) – Nozuko P. Blasich, Lindi M. Coetzee, Charlotte Sriruttan, Daniel DeSanto, Gregory S. Greene, Deborah K. Glencross, Nelesh P. Govender

 

  1. Association of Semi-Quantitative Cryptococcal Antigen Results in Plasma with Subclinical Cryptococcal Meningitis and Mortality Among Patients with Advanced HIV Disease (2021) – Nozuko P. Blasich, Rachel M. Wake, Ivy Rukasha, Yvonne Prince, Nelesh P. Govender

 

  1. Cryptococcus neoformans: Diagnostic Dilemmas, Electron Microscopy and Capsular Variants (2018) – Nozuko P. Blasich, Monica Birkhead, Serisha D. Naicker, Ivy Rukasha, Juno Thomas, Charlotte Sriruttan, Shareef Abrahams, Grisselda S. Mavuso, Nelesh P. Govender

 

Anastasia Kovrizhina | Medicinal chemistry | Women Researcher Award

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Dr. Anastasia Kovrizhina | Medicinal chemistry | Women Researcher Award

PhD Reseracher, Tomsk Polytechnic University Russia

Anastasia Kovrizhina is a Russian researcher specializing in organic chemistry and biotechnology. She holds a Ph.D. from National Research Tomsk Polytechnic University, where she focuses on molecular modeling and the synthesis of biologically active compounds. Currently, she is a researcher at Tomsk Polytechnic University and serves as a scientist secretary. Her work includes the development of novel kinase inhibitors and fluorocarbon aza-heterocycles for anticancer treatments. She has been actively involved in international collaborations, including research internships at Montana State University, USA, and Novosibirsk Institute of Organic Chemistry, Russia. With an h-index of 7, she has published extensively in high-impact journals and has presented at numerous international and national conferences. She has received multiple prestigious scholarships and awards, including the Baden-Württemberg State Scholarship and the Government Scholarship of the Russian Federation. Her expertise spans chemical synthesis, biological assays, computational chemistry, and quantum calculations.

Profile

Scopus

Education 🎓

Anastasia Kovrizhina earned her Ph.D. (2019-2023) in Organic Chemistry from National Research Tomsk Polytechnic University, specializing in molecular modeling and drug synthesis. She completed her Master’s degree (2017-2019) in Biotechnology at the same institution, where she studied organic and applied chemistry. During her studies, she participated in an academic exchange at Karlsruhe Institute of Technology, Germany, where she took courses in bioinformatics, bioprocessing, and enzymology. She obtained her Bachelor’s degree (2013-2017) in Biotechnology from National Research Tomsk Polytechnic University, with a strong foundation in chemistry, physics, and humanities. Her academic journey has been complemented by advanced training in computational chemistry, quantum calculations, and SAR/QSAR analysis. She has also gained international exposure through scholarships and research projects focused on innovative drug development. Her multidisciplinary education allows her to integrate experimental and computational approaches for pharmaceutical and medical applications.

Experience 🧑‍🏫

Anastasia Kovrizhina is currently a researcher at Tomsk Polytechnic University, specializing in the synthesis of biologically active compounds. She also serves as a scientist secretary at the School of Advanced Manufacturing Technologies and is an active member of the Council of Young Scientists. She has undertaken research internships at the Novosibirsk Institute of Organic Chemistry (2020) and Montana State University, USA (2019), where she collaborated on immunology and organic chemistry projects. Her work includes grant-funded research on kinase inhibitors, fluorocarbon aza-heterocycles, and polymer scaffolds for cardiovascular applications. She has supervised undergraduate and master’s students and has taught courses in professional English and organic chemistry. Her expertise includes molecular modeling, chemical synthesis, and computational chemistry. She has contributed to multiple research projects under the Russian Science Foundation and has been instrumental in developing innovative drug delivery systems for anticancer treatments.

 Awards & Honors 🏆

Anastasia Kovrizhina has received several prestigious awards, including the First Degree Diploma (2024) for her research on indenoquinoxalinone oxime (IQ-1). She won the 5th All-Russian Research Competition (2020) for her work on indenoquinoxaline derivatives. She was honored with the 3rd Degree Medal for “Achievements for Tomsk Polytechnic University” and the BAYHOST Scholarship for studying German (2020). She received the Baden-Württemberg State Scholarship (2018-2019) and the Russian Government Scholarship (2018-2019). Her participation in international conferences has been recognized with numerous accolades. She has also secured multiple research grants, including the Russian Science Foundation grants for developing kinase inhibitors and fluorocarbon aza-heterocycles as anticancer agents. Her scientific contributions to drug discovery and pharmaceutical chemistry have positioned her as a promising young researcher in her field.

Research Interests 🔬

Anastasia Kovrizhina’s research focuses on the synthesis and molecular modeling of biologically active compounds, particularly kinase inhibitors and fluorocarbon aza-heterocycles for anticancer treatments. She has pioneered the development of JNK kinase inhibitors based on indenoquinoxaline scaffolds, which have potential anti-inflammatory applications. Her work has demonstrated that IQ-1 salts enhance the efficacy of cerebral ischemia treatment. She has conducted pharmacokinetic studies on IQ-1 absorption in the gastrointestinal tract to optimize drug formulation. Her expertise extends to computational chemistry, quantum calculations, and structure-activity relationship (SAR) studies. She is also involved in developing supramolecular complexes for innovative drug delivery. Her interdisciplinary approach integrates synthetic chemistry, computational modeling, and biological assays to advance pharmaceutical research. She has contributed significantly to drug design, molecular docking studies, and the synthesis of novel heterocyclic compounds for targeted therapies.

Publications 📚

  1. Title: 6,8-Dibromo-11H-indeno[1,2-b]quinolin-11-one
    Year: 2024
    Author: Anastasia R. Kovrizhina, Dauren Tolegen, Dmitry I. Pavlov, Andrei S. Potapov, Andrei I. Khlebnikov
    Citations: Not available
    Article: Molbank

 

  1. Title: Evaluation of Nitric Oxide-Donating Properties of 11H-indeno[1,2-b]quinoxalin-11-one Oxime (IQ-1) by Electron Paramagnetic Resonance Spectroscopy
    Year: 2024
    Author: Viacheslav V. Andrianov, Igor A. Schepetkin, Leah V. Bazan, Khalil L. Gainutdinov, Anastasia R. Kovrizhina, Dmitriy N. Atochin, Andrei I. Khlebnikov
    Citations: Not available
    Article: Molecules

 

  1. Title: Dose proportionality and bioavailability of quinoxaline-based JNK inhibitor after single oral and intravenous administration in rats
    Year: 2024
    Author: Galina A. Frelikh, Elena A. Yanovskaya, Alexander P. Lakeev, Galina A. Chernysheva, Vera I. Smolyakova, Anastasia R. Kovrizhina
    Citations: Not available
    Article: Xenobiotica

 

  1. Title: Neuroprotective Effects of Tryptanthrin-6-Oxime in a Rat Model of Transient Focal Cerebral Ischemia
    Year: 2023
    Author: Mark Plotnikov, Galina A. Chernysheva, Vera I. Smol’yakova, Oleg I. Aliev, Anna M. Anishchenko, Olga A. Ulyakhina, Eugene S. Trofimova, Anastasia A. Ligacheva, Nina D. Anfinogenova, Anton Osipenko et al.
    Citations: Not available
    Article: Pharmaceuticals

 

  1. Title: Novel Tryptanthrin Derivatives with Selectivity as c–Jun N–Terminal Kinase (JNK) 3 Inhibitors
    Year: 2023
    Author: Igor A. Schepetkin, Oleksander S. Karpenko, Anastasia R. Kovrizhina, Liliya N. Kirpotina, Andrei I. Khlebnikov, Stepan I. Chekal, Alevtyna V. Radudik, Maryna O. Shybinska, Mark T. Quinn
    Citations: Not available
    Article: Molecules

 

  1. Title: Quantification of a promising JNK inhibitor and nitrovasodilator IQ-1 and its major metabolite in rat plasma by LC–MS/MS
    Year: 2022
    Author: Alexander P. Lakeev, Galina A. Frelikh, Elena A. Yanovskaya, Anastasia R. Kovrizhina, Vladimir V. Udut
    Citations: Not available
    Article: Bioanalysis

 

  1. Title: Poly(ϵ-caprolactone) Scaffolds Doped with c-Jun N-terminal Kinase Inhibitors Modulate Phagocyte Activation
    Year: 2019
    Author: K.S. Stankevich, I.A. Schepetkin, S.I. Goreninskii, A.K. Lavrinenko, E.N. Bolbasov, A.R. Kovrizhina, L.N. Kirpotina, V.D. Filimonov, A.I. Khlebnikov, S.I. Tverdokhlebov et al.
    Citations: Not available
    Article: ACS Biomaterials Science and Engineering

 

JAYAPRAKASH BEHERA| Medicinal chemistry | Young Scientist Award

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Mr. JAYAPRAKASH BEHERA| Medicinal chemistry | Young Scientist Award

Research scholar, CSIR-IIIM JAMMU, India

Jayaprakash Behera, an emerging researcher in Chemistry and Materials Science, holds a PhD from CSIR-IIIM Jammu under AcSIR. He is currently a Project Associate for CSIR Aroma Mission Phase-III. With a background in Polymer Chemistry and Organic Chemistry, he has worked on various research projects at prestigious institutions like IIT Guwahati and IIT Delhi. His innovative research has earned him multiple national and international accolades, including world records and recognition for contributions in scientific development.

Publication Profile

Scholar

🎓 Education 

PhD: CSIR – IIIM Jammu (continuing). M.Phil. Polymer Chemistry & Material Science, Veer Surendra Sai University of Technology (2020). M.Sc. Organic Chemistry, Galgotias University (2017). B.Sc. Chemistry, BJB Autonomous College, Utkal University (2013)

💼 Experience 

Jayaprakash has served as Project Associate for CSIR Aroma Mission Phase-III (2023–present) and Phase-II (2021–2023). He worked as JRF in a DST-funded project at Malaviya National Institute of Technology (2017-2019) and undertook major and minor projects at IIT Delhi and IIT Guwahati. He has also contributed significantly to national and international exhibitions and research projects on medicinal and nano-based products.

🏆 Awards & Honors 

Jayaprakash has received multiple prestigious awards, including the Dr. A.P.J. Abdul Kalam National Star Award, Young Scientist Award, City Excellence Award, Global Icon Award, and Rabindranath Tagore Hall of Fame Award. He is also a five-time world record holder, recognized by the London Book of World Records, USA Book of World Records, and more. Additionally, he has received accolades for his innovative ideas and contributions from CSIR and other organizations.

🔬 Research Focus 

Jayaprakash’s research revolves around Polymer Chemistry, Materials Science, and Nanotechnology, focusing on skin and hair-related solutions, nanoparticle seed coatings, and medicinal products. His work includes nano formulations for agricultural use, innovative medicinal soaps for skin issues, and skin and hair care solutions. He has authored multiple international articles and patents on his discoveries, contributing to the advancement of green chemistry and sustainable material science.

Publication Top Notes

  1. Nano boron nitride laminated poly (ethyl methacrylate)/poly (vinyl alcohol) composite films imprinted with silver nanoparticles as gas barrier and bacteria resistant packaging
    • Year: 2024
    • Authors: J Behera, S Patra, S Nazrul, SK Sharma, D Kumar, MK Verma, AK Katare, …
    • Citations: 2

 

  1. Bioassay-guided fractionations of Cannabis sativa extract and HPLC-assisted purifications of anti-proliferative active fractions lead to the isolation of 16 known and …
    • Year: 2024
    • Authors: Y Nalli, S Bharti, T Amin, R Singh, J Behera, SS Bhayye, YP Bharitkar, …
    • Citations: 2

 

  1. Correction: Bioassay-guided fractionations of Cannabis sativa extract and HPLC-assisted purifications of anti-proliferative active fractions lead to the isolation of 16 known …
    • Year: 2024
    • Authors: Y Nalli, S Bharti, T Amin, R Singh, J Behera, SS Bhayye, YP Bharitkar, …

 

  1. Phytochemical investigation of anti-proliferative active fractions of Cannabis sativa leads to isolate a new Compound Canniprene A and other bioactive compounds through …
    • Year: 2023
    • Authors: Y Nalli, S Bharti, T Amin, R Singh, J Behera, A Goswami, MK Verma

Antonios Kousaxidis | Medicinal Chemistry | Best Researcher Award

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 Mr. Antonios Kousaxidis | Medicinal Chemistry |Best Researcher Award

 Mr at School of Pharmacy, Aristotle University of Thessaloniki, Greece

A seasoned educator and researcher with extensive experience in physics, holding positions from Assistant to Associate Professor at IAU, Urmia, and Urmia University of Technology. Specialized in teaching a range of undergraduate to Ph.D. courses including Quantum Mechanics, Laser Physics, and Nonlinear Dynamical Systems. Proficient in Maple and Matlab programming with a strong background in finite element method analysis. Led impactful research projects in chaotic systems, cancer treatment, and national security, earning multiple awards including the Kharazmi Scientific Festival Second Prize. A recognized leader in academia with a commitment to advancing scientific knowledge and education.

Profile

  1. Scopus

🎓 Education:

Master’s Degree in Medicinal Chemistry: (9.85/10) from Departments of Chemistry, Medicine, Biological Applications and Technology, University of Ioannina, 45110, Ioannina, Greece. Bachelor’s Degree in Chemistry: (7.76/10) from Department of Chemistry, School of Sciences, University of Ioannina, 45110, Ioannina, Greece.

Personal Skills:

Synthetic Organic Chemistry and Biochemistry: Training in synthetic organic chemistry and biochemistry applied to drug design, with experience in several areas of synthetic methodology using retrosynthetic approaches. Metal-Based Coupling Reactions: Excellent knowledge and practice of metal-based coupling reactions in modern organic chemistry. Synthetic Routes Optimization: Training in synthetic routes optimization using one-pot reactions during master’s thesis. Analytical Methods: Proficient in NMR, IR, UV, and mass spectrometry for identifying organic compounds. Small Molecule Synthesis: Synthesis of small molecule organic compounds and isolation by recrystallization. Purification and Separation: Excellent knowledge and practice in chromatographic methods like column, preparative, and thin-layer chromatography for purifying and separating organic compounds. Biochemical Protocols: Good practice in using biochemical protocols for enzyme kinetics experiments. Drug Discovery Programs: Extensive experience in drug discovery programs, structure-based drug design, molecular docking, and SAR estimation models using in silico methods (Discovery Studio, Chimera, LigandScout, PyMOL, OpenBabel, ADMET). Scientific Manuscripts: Proficient in writing and preparing scientific manuscripts.

💻 Software Skills:

Office Suite (ECDL degree) – Word processing, spreadsheets, presentations, etc. Calculative and predictive programs like MestReNova, Topspin DataAnalysis, ChemDraw Ultra, MedChem Designer, and BioLoom.

Research Focus:

A. Kousaxidis primarily focuses on the design and synthesis of novel compounds with therapeutic potential, particularly targeting enzymes such as aldose reductase (ALR2) and protein tyrosine phosphatase 1B (PTP1B). The research also encompasses antimicrobial agents, lipoxygenase inhibitors, and therapeutic strategies for conditions like diabetes mellitus and sepsis.

Publications Top Notes 📝

  • A Molecular Hybridization Approach for the Design of Selective Aldose Reductase (ALR2) Inhibitors and Exploration of Their Activities Against Protein Tyrosine Phosphatase 1B (PTP1B)
    • Authors: Kousaxidis, A., Petrou, A., Rouvim, P., Nicolaou, I., Geronikaki, A.
    • Journal: Journal of Molecular Structure
    • Year: 2023
    • Volume: 1271
    • Article Number: 134116
    • Citations: 3
    • Summary: This study presents a hybridization approach to develop selective ALR2 inhibitors and investigates their potential activities against PTP1B, highlighting their dual therapeutic potential.

 

  • Design, Synthesis, and Pharmacological Evaluation of Indazole Carboxamides of N-Substituted Pyrrole Derivatives as Soybean Lipoxygenase Inhibitors
    • Authors: Lavrentaki, V., Kousaxidis, A., Theodosis-Nobelos, P., Koutsopoulos, K., Nicolaou, I.
    • Journal: Molecular Diversity
    • Year: 2023
    • Citations: 2
    • Summary: This paper discusses the synthesis and evaluation of novel indazole carboxamides, demonstrating significant inhibitory activity against soybean lipoxygenase.

 

  • N-Derivatives of (Z)-Methyl 3-(4-Oxo-2-thioxothiazolidin-5-ylidene)methyl)-1H-indole-2-carboxylates as Antimicrobial Agents—In Silico and In Vitro Evaluation
    • Authors: Petrou, A., Geronikaki, A., Kartsev, V., Nicolaou, I., Vizirianakis, I.S.
    • Journal: Pharmaceuticals
    • Year: 2023
    • Volume: 16
    • Issue: 1
    • Article Number: 131
    • Citations: 4
    • Summary: This open-access article evaluates the antimicrobial activity of new N-derivatives, supported by both in silico and in vitro methods.

 

  • Non-acidic Bifunctional Benzothiazole-Based Thiazolidinones with Antimicrobial and Aldose Reductase Inhibitory Activity as a Promising Therapeutic Strategy for Sepsis
    • Authors: Kousaxidis, A., Kovacikova, L., Nicolaou, I., Stefek, M., Geronikaki, A.
    • Journal: Medicinal Chemistry Research
    • Year: 2021
    • Volume: 30
    • Issue: 10
    • Pages: 1837-1848
    • Citations: 13
    • Summary: This research explores benzothiazole-based thiazolidinones with dual activity, suggesting a promising approach for treating sepsis.

 

  • Aldose Reductase and Protein Tyrosine Phosphatase 1B Inhibitors as a Promising Therapeutic Approach for Diabetes Mellitus
    • Authors: Kousaxidis, A., Petrou, A., Lavrentaki, V., Nicolaou, I., Geronikaki, A.
    • Journal: European Journal of Medicinal Chemistry
    • Year: 2020
    • Volume: 207
    • Article Number: 112742
    • Citations: 39
    • Summary: This review highlights the potential of targeting ALR2 and PTP1B as a therapeutic strategy for diabetes, emphasizing recent advances and future perspectives.

 

Simone Giovannuzzi | Medicinal chemistry | Young Scientist Award

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 Dr . Simone Giovannuzzi | Medicinal chemistry | Young Scientist Award

👨‍🏫Profile Summary

Dedicated researcher with a strong academic background in Pharmaceutical Sciences, specializing in drug development and computational chemistry. Recently awarded a PhD in Advanced Materials and Data Science, with expertise in multi-scale modeling and simulation of composite materials. Proficient in implementing computational methods and artificial intelligence models to advance pharmaceutical research. Fluent in English, French, and Arabic.

🌐 Professional Profiles

  1. Scopus Profile

 

  1. Orcid Profile

 

🎓 Education

PhD cum laude in Area del Farmaco e Trattamenti Innovativi: Curriculum Scienze Farmaceutiche NEUROFARBA Department, University of Florence, Italy Nov 2020 – Oct 2023 Qualification to practise the profession of Pharmacist National exam for professional qualification Jul 2020 5-year single-cycle Master’s Degree in Pharmaceutical Chemistry and Technologies Faculty of Pharmacy, University of Florence, Italy
Oct 2015 – Jun 2020

🔬Work Experience

Post-Doctoral Researcher in Area del Farmaco NEUROFARBA Department, University of Florence, Italy Nov 2023 – Present Tutor Senior in Area del Farmaco PNRR Plan “Orientamento attivo nella transizione scuola-Università”, Next Generation EU programme (NGEU) Oct 2023 – Present Tutor In-itinere for Chemistry, Organic Chemistry and Spectroscopic Methods Scuola di Scienze della Salute Umana, Corso di Scienze Farmaceutiche Applicate – Controllo Qualità (SFA-CQ), University of Florence, Italy Mar 2021 – Dec 2023 Internship Centre National de la Recherche Scientifique (CNRS), Montpellier, Occitanie, France Feb 2022 – Jul 2022

🔬Reviewer

Reviewer for international peer-reviewed scientific journals with high impact factor: Expert opinion on Therapeutic Patent Journal of Enzyme Inhibition and Medicinal Chemistry Frontiers Molecules Future Medicinal Chemistry Journal of the Turkish Chemical Society, Section A

🤝Major Ongoing Collaborations

Prof. J.Y. Winum, CNRS Montpellier, France, Prof. C. Capasso, CNR Napoli, Italy, Prof. G. De Simone, CNR Napoli, Italy, Prof. A.B. Vermelho, U. di Rio de Janeiro, Brazil, Prof. A. Aspatwar, U. Di Tampere, Finland, Prof. M. Bucciantini, U. Di Firenze, Italy, Prof. A. Ligresti, ICB Napoli, Italy Prof. F. Borges, U. di Porto, Portugal, Prof. Daniel P. Flaherty, U. di Purdue, USA, Mohamed N. Seleem, U. della Virgina, USA, Prof. S. Carradori, U. di Chieti, Italy

🧠Personal Skills

Excellent collaboration and coaching skills within a team, Outstanding problem-solving abilities, Strong adaptability and flexibility, Excellent active listening skills, Excellent creativity, Strong inclination towards research, Excellent multitasking and time management skills

💻Technical Skills

NMR, IR Spectroscopy, UV-Vis and Fluorescence Absorption, Multi-Step synthesis, Structure-Activity Relationship (SAR) Studies, Stopped-Flow Technique, Literature Review and Patent Analysis

🖥️Digital Skills

ChemDraw, SciFinder, Reaxys, Topspin, Origin, MestReNova, MS Office, E-Learning Platform, AI tools (ChatGPT, Perplexity)

📚Top Noted Publication

  1. Year: 2022
    • Journal: Composite Structure Journal
    • Title: Multiparametric modeling of composite materials based on non-intrusive PGD informed by multiscale analyses: Application for real-time stiffness prediction of woven composites.

 

  1. Year: 2023
    • Journal: Journal of the Mechanics and Physics of Solids
    • Title: Multiscale Thermodynamics-Informed Neural Networks (MuTINN) towards Fast and Frugal Inelastic Computation of Woven Composite Structures.

 

  1. Year: 2023 (under process)
    • Journal: Composite Structure Journal
    • Title: Multiparametric modeling of composite materials based on non-intrusive PGD informed by multiscale analyses: Application for real-time virtual testing of woven composites.